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Search Results for " dopamine beta-hydroxylase "
Targets Recommended: Others

11

抑制剂 & 化合物

4

天然产物

1

重组蛋白

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Cat. No. Product Name Target Signaling Pathways
T19654 Guanoclor

胍氯酚,VATENSOL

Others Others
Guanoclor (VATENSOL) 也称为guanochlor,是一种交感神经药物。已知它与猪肾膜中的非肾上腺素能位点结合。
T13383 Zamicastat

BIA 5-1058

BCRP; Hydroxylase; P-gp Membrane transporter/Ion channel; Metabolism; Neuroscience
Zamicastat (BIA 5-1058) 是多巴胺 β-羟化酶 (DBH) 抑制剂,可透过血脑屏障引起中枢和周边效应,具有降血压作用。它也是一种浓度依赖性的双重 P-gp 和 BCRP 抑制剂,IC50值分别为 73.8 和 17.0 μM。
T6604 Nepicastat hydrochloride

Nepicastat HCl,内匹司他盐酸盐,RS-25560-197 hydrochloride,SYN-117 hydrochloride,Nepicastat (SYN-117) HCl

Hydroxylase Metabolism
Nepicastat hydrochloride (RS-25560-197 hydrochloride) 是一种选择性的,有效的,口服活性的多巴胺 β 羟化酶(dopamine-beta-hydroxylase)抑制剂,对牛和人多巴胺 β 羟化酶的IC50分别为IC50=8.5 nM 和IC50=9 nM。Nepicastat HCl 可以穿过血脑屏障。
T30615 Bupicomide

Hydroxylase Metabolism
Bupicomide 是一种多巴胺β羟化酶抑制剂,具有抗高血压和血管扩张活性,可降低14C-多巴胺的14C-去甲肾上腺素生物合成,可用于研究高血压。
T11238L Etamicastat hydrochloride

BIA 5-453 hydrochloride

Dehydrogenase Metabolism
Etamicastat hydrochloride (BIA 5-453 hydrochloride) 是一种外周选择性多巴胺β-羟化酶抑制剂,具有降低高血压的作用。
T50049 4-Methylhistamine hydrochloride

Others Others
4-Methylhistamine hydrochloride 已被证明能抑制铜依赖性酶如酪氨酸酶和多巴胺β-羟化酶的活性,还被证明可以调节参与细胞周期调节和凋亡的基因的表达。
T71936 Phenylthiazolylthiourea

Phenylthiazolylthiourea ia a dopamine-beta-hydroxylase inhibitor.
T69568 FLA-63

FLA-63 is a dopamine-beta-hydroxylase (DBH)-inhibitor and an inhibitor of the last step of noradrenaline biosynthesis.
T23848 Calcium Fusarate

Calcium Fumarate is an inhibitor of dopamine beta-hydroxylase. It also inhibited cell proliferation and DNA synthesis.
T70209 Nepicastat hydrochloride monohydrate

Nepicastat hydrochloride monohydrate is an inhibitor of dopamine beta-hydroxylase, an enzyme that catalyzes the conversion of dopamine to norepinephrine.
T60633 Nepicastat

Nepicastat (SYN117) 是一种选择性的,有效的,口服的多巴胺 β 羟化酶抑制剂,可穿过血脑屏障(BBB)。Nepicastat (SYN117) 对牛和人多巴胺 β 羟化酶产生浓度依赖性抑制作用,IC50值分别为8.5 nM 和 9 nM。

化合物

Guanoclor
Cat.No: T19654
Synonym: 胍氯酚,VATENSOL
Target: Others
Zamicastat
Cat.No: T13383
Synonym: BIA 5-1058
Target: BCRP, Hydroxylase, P-gp
Nepicastat hydrochloride
Cat.No: T6604
Synonym: Nepicastat HCl,内匹司他盐酸盐,RS-25560-197 hydrochloride,SYN-117 hydrochloride,Nepicastat (SYN-117) HCl
Target: Hydroxylase
Bupicomide
Cat.No: T30615
Synonym:
Target: Hydroxylase
Etamicastat hydrochloride
Cat.No: T11238L
Synonym: BIA 5-453 hydrochloride
Target: Dehydrogenase
4-Methylhistamine hydrochloride
Cat.No: T50049
Synonym:
Target: Others
Phenylthiazolylthiourea
Cat.No: T71936
Synonym:
Target:
FLA-63
Cat.No: T69568
Synonym:
Target:
Calcium Fusarate
Cat.No: T23848
Synonym:
Target:
Nepicastat hydrochloride monohydrate
Cat.No: T70209
Synonym:
Target:
Nepicastat
Cat.No: T60633
Synonym:
Target:
Cat. No. Product Name Target Signaling Pathways
T6S0923 Hypericin

Hypericine,金丝桃素,Cyclosan

Apoptosis; Antiviral; Influenza Virus; Tyrosine Kinases; Antibacterial; PKC Apoptosis; Chromatin/Epigenetic; Cytoskeletal Signaling; Immunology/Inflammation; Microbiology/Virology; Tyrosine Kinase/Adaptors
Hypericin (Cyclosan) 是贯叶连翘的提取物,有抗菌、抗病毒、抗肿瘤和抗抑郁作用。
T2S1778 DL-Goitrin

DL-甲状腺肿素,板蓝根,Goitrin,(R,S)-告依春

Others Others
DL-Goitrin 也称为 (R,S)-Goitrin,由 epigoitrin (R-Goitrin) 和告依春 (S-Goitrin) 两种异构体组成,是板蓝根的成分。
TN2252 Syrosingopine

Dopamine Receptor GPCR/G Protein; Neuroscience
Syrosingopine 是 MCT1和 MCT4双重抑制剂,对 MCT4 的效力高 60 倍,可防止乳酸和 H+ 流出。它是可口服抗高血压药物,联合二甲双胍具有研究癌症疾病的潜力。
T25900 Oosponol

Lenzitin

Oosponol is a dopamine beta-hydroxylase inhibitor exhibiting hypotensive effects.

天然产物

Hypericin
Cat.No: T6S0923
Synonym: Hypericine,金丝桃素,Cyclosan
Target: Apoptosis, Antiviral, Influenza Virus, Tyrosine Kinases, Antibacterial, PKC
DL-Goitrin
Cat.No: T2S1778
Synonym: DL-甲状腺肿素,板蓝根,Goitrin,(R,S)-告依春
Target: Others
Syrosingopine
Cat.No: TN2252
Synonym:
Target: Dopamine Receptor
Oosponol
Cat.No: T25900
Synonym: Lenzitin
Target:
Cat. No. Product Name Species Expression System
TMPY-03852 Dopamine beta-Hydroxylase Protein, Human, Recombinant (His)

dopamine β-hydroxylase (dopamine ...

Human HEK293 Cells
DBH is a 29 kDa copper-containing oxygenase. It can be detected in noradrenergic nerve terminals of the central and peripheral nervous systems, and is also expressed in chromaffin cells of the adrenal medulla. DBH contains our identical subunits, and its activity requires ascorbate as a cofactor. It functions in in the synthesis of small-molecule neurotransmitters that is membrane-bound, making norepinephrine the only transmitter synthesized inside vesicles. DBH has been shown to be associated ...

重组蛋白

Dopamine beta-Hydroxylase Protein, Human, Recombinant (His)
Cat.No: TMPY-03852
Species: Human
Expression System: HEK293 Cells
TargetMol Loading
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